Open access peer-reviewed Edited Volume


Synthesis and Biological Activities


Sadashiv S. O.

Garden City University

Heterocycles have constituted the largest area of research in organic chemistry. These heterocycles play an important role in biochemical processes because the side groups of the most typical and essential constituents of living cells, DNA and RNA, are based on aromatic heterocycles. Many synthetic methods have been developed for the preparation of heterocycles. The recent surge of interest in the chemistry of heterocycles can be explained by their unusual properties and exotic structure. These heterocycles include highly stable aromatic compounds that display physicochemical properties with relevance in the design of new materials. Thus, heterocycles contribute to the development of society from a biological and industrial point of view.

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HeterocyclesSynthesis and Biological ActivitiesEdited by Belakatte Parameshwarappa Nandeshwarappa

Published: June 10th 2020

DOI: 10.5772/intechopen.78709

ISBN: 978-1-83880-624-8

Print ISBN: 978-1-83969-003-7

eBook (PDF) ISBN: 978-1-83880-625-5

Copyright year: 2020

Books open for chapter submissions

7157 Total Chapter Downloads

13 Crossref Citations

1 Web of Science Citations

19 Dimensions Citations


Open access peer-reviewed

1. Introductory Chapter: Synthesis and Antimicrobial Activities of Dihydroazeto[2′,3′:4,5]seleno[2,3-b]quinolines

By B.P. Nandeshwarappa, G.K. Prakash and S.O. Sadashiv


Open access peer-reviewed

2. Phenacyl Bromide: An Organic Intermediate for Synthesis of Five- and Six-Membered Bioactive Heterocycles

By Dinesh Kumar Jangid and Surbhi Dhadda


Open access peer-reviewed

3. Amidoxime Derivatives with Local Anesthetic, Antitubercular, and Antidiabetic Activity

By Lyudmila Kayukova, Umirzak Jussipbekov and Kaldybay Praliyev


Open access peer-reviewed

4. Recent Developments of Target-Based Benzimidazole Derivatives as Potential Anticancer Agents

By Nerella Sridhar Goud, Pardeep Kumar and Rose Dawn Bharath


Open access peer-reviewed

5. Thiazole Moiety: An Interesting Scaffold for Developing New Antitumoral Compounds

By Sandra Ramos-Inza, Carlos Aydillo, Carmen Sanmartín and Daniel Plano


Open access peer-reviewed

6. One-Pot-Condensation Reaction of Heterocyclic Amine, 1,3-Diketone and Aldehydes Using In Situ Generated Superoxide Ion: A Rapid Synthesis of Structurally Diverse Drug-Like Complex Heterocycles

By Sundaram Singh and Savita Kumari


Open access peer-reviewed

7. The Oxygen-Containing Fused Heterocyclic Compounds

By Hillemane Venkatachalam and Nanjangud Venkatesh Anil Kumar


Open access peer-reviewed

8. Synthesis and Anticancer Evaluation of Benzenesulfonamide Derivatives

By Dattatraya Navnath Pansare and Rohini Narayan Shelke


Open access peer-reviewed

9. Synthesis and Biological Evaluation of Novel Phosphonyl Thiazolo Pyrazoles

By Avula Srinivas


Open access peer-reviewed

10. Quinoline Heterocycles: Synthesis and Bioactivity

By Yamajala B.R.D. Rajesh


Open access peer-reviewed

11. Potent Antibacterial Profile of 5-Oxo-Imidazolines in the New Millennium

By Roshan D. Nasare, Mohammad Idrees, Satish S. Kola and Rajendra S. Dongre


Open access peer-reviewed

12. Azoles as Potent Antimicrobial Agents

By Rohit Singh and Swastika Ganguly


Edited Volume and chapters are indexed in

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  • Google Scholar
  • AZ ebsco
  • Base
  • CNKI

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